Page last updated: 2024-09-04

celastrol methyl ester and (1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol

celastrol methyl ester has been researched along with (1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol in 1 studies

Compound Research Comparison

Studies
(celastrol methyl ester)
Trials
(celastrol methyl ester)
Recent Studies (post-2010)
(celastrol methyl ester)
Studies
((1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol)
Trials
((1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol)
Recent Studies (post-2010) ((1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol)
3902717012

Protein Interaction Comparison

ProteinTaxonomycelastrol methyl ester (IC50)(1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol (IC50)
XBP1Homo sapiens (human)4.76
DNA damage-inducible transcript 3 proteinMus musculus (house mouse)2.53
Epidermal growth factor receptorHomo sapiens (human)0.7944
Tyrosine-protein kinase FynHomo sapiens (human)0.7221
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)1.4004
Muscarinic acetylcholine receptor M4Homo sapiens (human)4.561
Muscarinic acetylcholine receptor M5Homo sapiens (human)4.4868
Alpha-2A adrenergic receptorHomo sapiens (human)2.0232
Adenosine receptor A3Homo sapiens (human)3.7058
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.505
Beta-3 adrenergic receptorHomo sapiens (human)4.9963
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)3.7058
Alpha-2C adrenergic receptorHomo sapiens (human)3.446
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.5435
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.6238
Substance-K receptorHomo sapiens (human)6.7929
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.4004
Histamine H2 receptorHomo sapiens (human)0.1081
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.5435
Sodium-dependent serotonin transporterHomo sapiens (human)1.2532
Histamine H1 receptorHomo sapiens (human)5.1768
D(3) dopamine receptorHomo sapiens (human)2.1039
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.939
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)3.7058
Sodium-dependent dopamine transporter Homo sapiens (human)2.57
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.1172

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y1

Other Studies

1 other study(ies) available for celastrol methyl ester and (1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol

ArticleYear
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
    Science (New York, N.Y.), 2011, Dec-09, Volume: 334, Issue:6061

    Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites

2011